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I.Scientific
papers
II.Proceedings
III.Conference communications
IV.Invited speakers
V.Chairpersons
VI.Awards
VII.Visiting researchers
VIII.Visiting students
I. Scientific
papers
-
C. Padula, A. Fulgoni, P. Santi.
“In vivo stratum corneum
distribution of lidocaine, assessed by tape stripping,
from a new bioadhesive film”, Skin
Research and Technology, 16,
125-130 (2010).
-
M. Fantini, V. Zuliani, M.A. Spotti,
M. Rivara. “Microwave assisted
efficient synthesis of imidazolo-based privileged
structures”, Journal of
Combinatorial Chemistry, 12,
181-185 (2010).
-
M.C. Rodríguez-Argüelles,
S. Mosquera-Vázquez, Jesús Sanmartín-Matalobos, A.M.
García-Deibe, C. Pelizzi, F. Zani.
“Evaluation of the antimicrobial activity of some chloro
complexes of imidazolo-2-carbaldehyde semicarbazone:
X-ray crystal structure of cis-NiCl2(H2L)(H2O)”,
Polyhedron,
29, 864-870 (2010).
-
Y. Gerelli, M.T. Di Bari, S.
Barbieri, F. Sonvico, P. Colombo, F. Natali, A. Deriu.
“Flexibility and drug release
features of lipid/saccaride nanoparticles”,
Soft Matter,
6, 685-691 (2010).
-
R. Bettini, R. Menabeni, R. Tozzi,
M.B. Pranzo, I. PasqualI, M.R. Chierotti, R. Gobetto, L.
Pellegrino. “Didanosine
polymorphism in a supercritical antisolvent process”,
Journal of Pharmaceutical Sciences,
99(4), 1855-1870 (2010).
-
C.
Balaguer-Fernández, C. Padula, A. Femenía-Font, V.
Merino, P. Santi, A. López-Castellano.
“Development and evaluation of occlusive systems
employing polyvinyl alcohol for transdermal delivery of
sumatriptan succinate”, Drug
Delivery, 17(2),
83-91 (2010).
-
T.T.N. Huynh, K.
Padois, F. Sonvico, A. Rossi, F. Zani, F. Pirot, J.
Doury, F. Falson.
“Characterization of a polyuretane-based controller
release system for local delivery of chlorhexidine
diacetate”, European Journal of
Pharmaceutics and Biopharmaceutics,
74, 255-264 (2010).
-
R.P. Raffin, L.
Colomé, C.R.D. Hoffmeister, P. Colombo, A. Rossi, F.
Sonvico, L.M. Colomé, C.C. Natalini, A.R. Pohlmann, T.
Dalla Costa, S.S. Guterres.
“Pharmacokinetics evaluation of soft agglomerates for
prompt delivery of enteric pantoprazole-loaded
microparticles”, European Journal
of Pharmaceutics and Biopharmaceutics,
74, 275-280 (2010).
-
L. Ampollini, F. Sonvico, E.
Barocelli, A. Cavazzoni, R. Bilancia, C. Mucchino, A.M.
Cantoni, P. Carbognani. “Intrapleural polymeric
films containing cisplatin for malignant pleural
mesotelioma in a rat tumour model: a preliminary study”,
European Journal of
Cardio-thoracic Surgery, 37,
557-565 (2010).
-
C. Carmi, A. Cavazzoni, S. Vezzosi,
F. Bordi, F. Vacondio, C. Silva, S. Rivara, A. Lodola,
R.R. Alfieri, S. La Monica, M. Galetti, A. Ardizzoni,
P.G. Petronini, M. Mor. “Novel
irreversibile epidermal growth factor receptor
inhibitors by chimica modulation of the cysteine-trap
portion”, Journal of Medicinal
Chemistry,
53, 2038-2050 (2010).
-
T. Şenyiğit, F. Sonvico, S.
Barbieri, Ö. Özer, P. Santi, P. Colombo.
“Lecithin/chitosan nanoparticles of
clobetasol-17-propionate capable of accumulation in pig
skin”, Journal of Controlled
Release, 142, 368-373
(2010).
-
L. Auzzas, F. Zanardi, L.
Battistini, P. Burreddu, P. Carta, G. Rassu, C. Curti,
G. Casiraghi. “Targeting
αvβ3
integrin: design and applications of multifunctional RGD-based
peptides and semipeptides”,
Current Medicinal Chemistry,
17, 1255-1299 (2010).
-
M. Casas, O.L.
Strusi, M.R. Jiménez-Castellanos, P. Colombo.
“Tapioca starch graft copolymers and Dome Matrix®
modules assembling technology. I. Effect of module shape
on drug release”, European Journal
of Pharmaceutics and Biopharmaceutics,
75,
42-47 (2010).
-
V. Zambrano, G. Rassu, A. Roggio,
L. Pinna, F. Zanardi, C. Curti, G. Casiraghi, L.
Battistini. “Asymmetric total synthesis of
1-deoxy-7,8-di-epi-castanospermine”,
Organic & Biomolecular Chemistry,
8, 1725-1730 (2010).
-
M. Rivara, M. Fantini, D. Acquotti,
V. Zuliani. “NMR analysis of a
series of imidazobenzoxazines”,
Magnetic Resonance in Chemistry,
48, 500-503 (2010).
-
M. Galetti, R.R. Alfieri, A.
Cavazzoni, S. La Monica, M. Bonelli, C. Fumarola, P.
Mozzoni, G. De Palma, R. Andreoli, A. Mutti, M. Mor, M.
Tiseo, A. Ardizzoni, P.G. Petronini.
“Funcional characterization of
gefitinib uptake in non-small cell lung cancer cell
lines”, Biochemical Pharmacology,
80, 179-187 (2010).
-
V. Zuliani, M. Rivara, M. Fantini,
G. Costantino. “Sodium channel
blockers for neuropathic pain”,
Expert Opinion on Therapeutic Patents,
20(6), 755-779 (2010).
-
O.L. Strusi, P. Barata, D. Traini,
P.M. Young, S. Mercuri, G. Colombo, F. Sonvico, R.
Bettini, P. Colombo.
“Artesunate-clindamycin multi-kinetics and site-specific
oral delivery system for antimalaric combination
products”, Journal of Controlled
Release, 146, 54-60
(2010).
-
F. Zanardi, L. Battistini, C. Curti,
G. Casiraghi, G. Rassu. “The
vinylogous aldol reaction: targeting stereocontrol”,
Chemtracts-Organic Chemistry,
23, 123-140 (2010).
-
L. Battistini, F. Zanardi, C. Curti,
G. Casiraghi. “The vinylogous
Mannich reaction: an asymmetric journey”,
Chemtracts-Organic Chemistry,
23, 141-152 (2010).
-
S. Nicoli, M. Eeman, M. Deleu, E.
Bresciani, C. Padula, P. Santi.
“Effect of lipopeptides and
iontophoresis on aciclovir skin delivery”,
Journal of Pharmacy and
Pharmacology, 62,
702-708 (2010).
-
D.R. de Araujo,
C. Padula, C.M.S. Cereda, G.R. Tófoli, R.B. Brito jr.,
E. de Paula, S. Nicoli, P. Santi.
“Bioadhesive films containing benzocaine: correlation
between in vitro permeation and in vivo
local anesthetic effect”,
Pharmaceutical Research, 27,
1677-1686 (2010).
-
M. Incerti, L. Flammini, F. Saccani,
G. Morini, M. Comini, M. Coruzzi, E. Barocelli, V.
Ballabeni, S. Bertoni.
“Dual-acting drugs: an in vitro study of nonimidazole
histamine H3 receptor antagonists combining
anticholinesterase activity”,
ChemMedChem, 5,
1143-1149 (2010).
-
M.B. Pranzo, D.
Cruickshank, M. Coruzzi, M.R. Caira, R. Bettini.
“Enantiotropically related albendazole polymorphs”,
Journal of Phamaceutical Sciences,
99,
3731-3742 (2010).
-
M. Mor, S. Rivara, D. Pala, A.
Bedini, G. Spadoni, G. Tarzia.
“Recent advances in the development of melatonin MT1
and MT2 receptor agonists”,
Expert Opinion in Therapeutic
Patents, 20(8),
1059-1076 (2010).
-
S. Pescina, G. Ferrari, P. Govoni,
C. Macaluso, C. Padula, P. Santi, S. Nicoli.
“In-vitro permeation of bevacizumab
through human sclera: effect of iontophresis
application”, Journal of Pharmacy
and Pharmacology, 62,
1189-1194 (2010).
-
C. Solorzano, F. Antonietti, A.
Duranti, A. Tontini, S. Rivara, A. Lodola, F. Vacondio,
G. Tarzia, D. Piomelli, M. Mor. “Synthesis and
structure-activity relationships of N-(2-oxo-3-oxetanyl)amides
as N-acylethanolamine-hydrolyzing acid amidase
inhibitors”, Journal of Medicinal
Chemistry, 53,
5770-5781 (2010).
-
C. Curti, B. Ranieri, L.
Battistini, G. Rassu, V. Zambrano, G. Pelosi, G.
Casiraghi, F. Zanardi. “Catalytic, asymmetric
vinylogous Mukaiyama aldol reactions of pyrrole- and
furan-based dienoxy silanes: how the diene heteroatom
impacts stereocontrol”, Advanced
Synthesis & Catalysis, 352,
2011-2022 (2010).
-
S.A. Al-Trawneh, J.A. Zahra, M.R.
Kamal, M.M. El-Abadelah, F. Zani, M. Incerti, A.
Cavazzoni, R.R. Alfieri, P.G. Petronini, P. Vicini.
“Synthesis and biological evaluation
of tetracyclic fluoroquinolones as antibacterial and
anticancer agents”, Bioorganic &
Medicinal Chemistry, 18,
5873-5884 (2010).
-
A. Lodola, J.
Sirirak, N. Fey, S. Rivara, M. Mor, A.J. Mulholland.
“Structural fluctuations in enzyme-catalyzed reactions:
determinants of reactivity in Fatty Acid Amide Hydrolase
from multivariate statistical analysis of quantum
mechanics/molecular mechanics paths”,
Journal of Chemical Theory and
Computation, 6,
2948-2960 (2010).
-
C. Padula, C. Chiapponi, M.T.
Dibari, A. Deriu, F. Sonvico, S. Barbieri, J. Ollivier,
P. Santi. “Single layer
transdermal film containing lidocaine: water and
lidocaine mobility determined using neutron scattering”,
Journal of Pharmaceutical Sciences,
99(10), 4277-4284 (2010).
-
G. Spadoni, A. Bedini, S. Rivara,
M. Mor. “Melatonin receptor
agonists: new options for insomnia and depression
treatment”, CNS Neuroscience &
Therapeutics, 00, 1-9
(2010).
-
F. Vacondio, C.
Silva, M. Mor, B. Testa.
“Qualitative structure-metabolism relationships in the
hydrolysis of carbamates”, Drug
Metabolism Reviews, 42(4),
551-589 (2010).
-
J.R. Clapper, G.
Moreno-Sanz, R. Russo, A. Guijarro, F. Vacondio, A.
Duranti, A. Tontini, S. Sanchini, N.R. Sciolino, J.M.
Spradley, A.G. Hohmann, A. Calignano, M. Mor, G. Tarzia,
D. Piomelli.
“Anandamide suppresses pain initiation through a
peripheral endocannabinoid mechanism”,
Nature Neuroscience,
13(10), 1265-1270 (2010).
-
V. Zuliani, M. Fantini, A. Nigam,
J.P. Stables, M.K. Patel, M. Rivara.
“Anticonvulsant activity of 2,4(1H)-diarylimidazoles
in mice and rats acute seizure models”,
Bioorganic & Medicinal Chemistry,
18, 7957-7965 (2010).
-
C. Curti, L. Battistini, F.
Zanardi, G. Rassu, V. Zambrano, L. Pinna, G. Casiraghi.
“Uncatalyzed, diastereoselective vinylogous Mukaiyama
aldol reactions on aqueous media: pyrrole vs furan
2-silyloxy dienes”, Journal of
Organic Chemistry, 75,
8681-8684 (2010).
-
C.
Padula, C. Ferretti, S. Nicoli, P. Santi, “Combined
patch containing salicylic acid and nicotinamide: role
of drug interaction”,
Current Drug Delivery,
7,
415-420 (2010).
II. Proceedings
-
B. Forbes, P. Colombo, G.
Brambilla, M. Saunders, S.A. Jones, F. Buttini.
“Important considerations regarding the bioequivalence
of particles emitted from becolmetasone dipropionate
solution metered dosed inhalers”,
Respiratory Drug Delivery 2010,
Orlando (Florida, USA), April 25th-29th,
2010. (ISBN 1-933722-42-8, pp 609-613).
III.Conference communications
(C) = Oral Communication
(P) = Poster
-
P. Vicini, R.A. Al-Qawasmeh, J.A. Zahra,
F. Zani, M.M. El-Abadelah. “Discovery of a lead for
the development of novel heterocycle-fused fluoroquinolones”,
4th International
Symposium on Current Trends in Drug Discovery Research,
Lucknow (India), February, 17th-21st,
2010. (P)
-
S. Pescina, G. Ferrari, C.
Macaluso, P. Santi, S. Nicoli.
“Iontophoretic trans-scleral permeation of high molecular
weight compounds”, 4th
AItUN Annual Meeting: Innovation in Pharmaceutics: “a
glimpse” in the Biotech world, Naples (Italy),
February, 26th-27th, 2010. (C)
-
M. Miozzi, P. Colombo, F. Buttini.
“Ciprofloxacin spray-dried powder for
pulmonary administration”, 4th
AItUN Annual Meeting: Innovation in Pharmaceutics: “a
glimpse” in the Biotech world, Naples (Italy),
February, 26th-27th, 2010. (P)
-
S. Mercuri, F.G. Di Girolamo, A. Rossi,
O.L. Strusi, F. Sonvico, P. Colombo.
“Multi-drug and multi-kinetics modular
assembled system for the treatment of Parkinson disease”,
4th AItUN Annual Meeting:
Innovation in Pharmaceutics: “a glimpse” in the Biotech
world, Naples (Italy), February, 26th-27th,
2010. (P)
-
L. Marin, E. Cuoghi, P. Colombo, F.
Buttini. “The development of
insulin dry powder blended with smoothed lactose for
pulmonary administration”, 4th
AItUN Annual Meeting: Innovation in Pharmaceutics: “a
glimpse” in the Biotech world, Naples (Italy),
February, 26th-27th, 2010. (P)
-
A.G. Balducci, G. Colombo, F.
Bortolotti, P. Colombo, A. Rossi.
“Development of artemisinin -β
cyclodextrin complex agglomerates”,
4th AItUN Annual Meeting: Innovation in
Pharmaceutics: “a glimpse” in the Biotech world,
Naples (Italy), February, 26th-27th,
2010. (P)
-
M. Miozzi, F. Sonvico, P. Colombo, F.
Buttini. “Construction of ciprofloxacin dry
microparticles for lung infection treatment”,
7th World Meeting on
Pharmaceutics, Biopharmaceutics and Pharmaceutical
Technology, La Valletta (Malta), March, 8th-11th,
2010. (P)
-
T. Şenyiğit, F. Sonvico, S. Barbieri,
Ö. Özer, P. Santi, P. Colombo. “Preparation and
characterization of clobetasol-17-propionate loaded
lecithin-chitosan nanoparticles for topical use”,
7th World Meeting on
Pharmaceutics, Biopharmaceutics and Pharmaceutical
Technology, La Valletta (Malta), March, 8th-11th,
2010. (P)
-
F. Sonvico.
“Lecithin/chitosan nanosystems for the delivery of
lipophilic drugs”, One day seminar
on New advances in drug delivery systems, Penang
(Malaysia), May, 24th, 2010. (C)
-
A. Rossi.
“Agglomerates for malaria treatment in children”,
One day seminar on New advances in
drug delivery systems, Penang (Malaysia), May, 24th,
2010. (C)
-
A.G. Balducci, P. Colombo, N.A.K. Khan,
K.H. Yuen, E. Magosso, G. Colombo, A. Rossi.
“Development of artemisinin soft
agglomerates”, Pharmatech 2010,
International Conference and Exhibition on Pharmaceutical,
Nutraceutical and Cosmeceutical Technology, Kuala
Lumpur (Malaysia), May 25th-27th,
2010. (C)
-
F. Sonvico, L. Ampollini, A.
Rossi, P. Carbognani, P. Colombo. “Cisplatin-loaded
polymeric films for the intrapleural treatment of malignant
pleural mesotelioma”, Pharmatech
2010, International Conference and Exhibition on
Pharmaceutical, Nutraceutical and Cosmeceutical Technology,
Kuala Lumpur (Malaysia), May 25th-27th,
2010. (C)
-
G. Colombo, A. Rimessi, A. De Corcelli,
E. Menegatti, F. Bortolotti, F. Sonvico, P. Colombo.
“Combination of alginate and cells for
skin re generation”, Pharmatech
2010, International Conference and Exhibition on
Pharmaceutical, Nutraceutical and Cosmeceutical Technology,
Kuala Lumpur (Malaysia), May 25th-27th,
2010. (P)
-
P. Vicini, A. Geronikaki.
“Antinflammatory potential of benzothiazole and
benzisothiazole derivatives”, 6th
Eurasian Meeting on Heterocyclic Chemistry, Alicante
(Spain), June 30th – July 4th, 2010.
(C)
-
F. Sonvico, L. Ampollini, E.
Barocelli, A. Cavazzoni, C. Mucchino, P.G. Petronini, P.
Carbognani, P. Colombo. “Polysaccharide films: a drug
delivery platform for loco-regional therapy of malignant
pleural mesothelioma”, The 10th
International Conference of the International Mesothelioma
Interest Group IMIG2010, Kyoto (Japan), August, 31st,
September, 3rd, 2010. (C)
-
L. Ampollini, E. Barocelli, F.
Sonvico, P. Colombo, R. Bilancia, A. Cavazzoni, P.G.
Petronini, A. Cantoni, M. Rusca, P. Carbognani.
“Intrapleural application of polymeric films containing
cisplatin and pemetrexed in a rat tumour model of malignant
pleural mesotelioma”, The 10th
International Conference of the International Mesothelioma
Interest Group IMIG2010, Kyoto (Japan), August, 31st,
September, 3rd, 2010. (C)
-
M. Miozzi, E. Cuoghi, P. Colombo, F.
Buttini. “Smoothed lactose as a
carrier for insulin pulmonary delivery”,
Meeting on Lactose as a Carrier for
Inhalation Products, Parma (Italy), September, 26th-28th,
2010. (P)
-
L. Marin, F. Sonvico, G. Massimo, P.
Colombo, F. Buttini. “Flowability
and respirabilità of insulin dry powder blends for pulmonary
administration”, Meeting on Lactose
as a Carrier for Inhalation Products, Parma (Italy),
September, 26th-28th, 2010. (P)
-
A. Rossi. A.G. Balducci, G.
Corace, C. Cavallari, L. Rodriguez, P. Colombo.
“Preparation of gastroresistant mesalazine lipidic
microcapsules”, XVIII International
Conference on Bioencapsulation, Porto (Portugal),
October, 1st-2nd, 2010. (C)
-
L. Pezzini, F. Guida, R. Bettini.
“Diazepam-PEG solid dispersion: miscibilità and solid state
stability”, 2nd
Conference Innovation in Drug Delivery: from preformulation
to Development through innovative evaluation process,
Aix en Provence (France), October 3rd-6th,
2010. (P)
-
R. Menabeni, C. Scarpignato, R. Bettini.
“Interaction of sucralfate with an
anti-arthritic drug in aqueous solution”,
2nd Conference Innovation
in Drug Delivery: from preformulation to Development through
innovative evaluation process, Aix en Provence
(France), October 3rd-6th, 2010.
(P)
-
S. Mercuri, O.L. Strusi, F. Sonvico, A.
Rossi, P. Colombo. “Dome Matrix
modular assembled system for the treatment of Parkinson’s
disease”, 2nd Conference
Innovation in Drug Delivery: from preformulation to
Development through innovative evaluation process,
Aix en Provence (France), October 3rd-6th,
2010. (P)
-
T. Senyigit, F. Sonvico, S. Barbieri,
P. Santi, P. Colombo, O. Ozer. “In vivo assessment of
clobetasol propinate loaded lecithin-chitosan nanoparticles
for topical use”,
2nd Conference Innovation in
Drug Delivery: from preformulation to Development through
innovative evaluation process, Aix en Provence
(France), October 3rd-6th, 2010. (P)
-
L. Pozzetti, C. Padula, S. Nicoli, P.
Santi. “Mucoadhesive films for
gingival administration of lidocaine”,
2nd
Conference on “Innovation in drug delivery: from
preformulation to development through innovative evaluation
process”, Aix-en-Provence,
Francia, October 3th-6th, 2010. (P)
-
P. Bertuzzi, C. Padula, S. Nicoli, P.
Santi. “In vitro study of
cutaneous accumulation of local anesthetics from polymeric
film”, 2nd
Conference on “Innovation in drug delivery: from
preformulation to development through innovative evaluation
process”, Aix-en-Provence,
Francia, October 3th-6th, 2010. (P)
-
M. Tognolini, C. Giorgio, I.H. Mohamed,
L. Flammini, M. Incerti, A. Lodola, E. Barocelli.
“Lithocholic acid competitively inhibits
EphA2-ephrinA1 binding: pharmacological and structural
considerations”, Lost in
translation: bridging the gap between cancer research and
effective terapies, Rome (Italy), October 4th-7th,
2010. (Poster P04). (P)
-
J. Zahra, M.
El-Abadelah, S. Al-Trawneh, P. Vicini, F. Zani.
“Antibacterial activity of
tetracyclic fluoroquinolones with a
4-oxothieno[2’,3’:4,5]pyrrolo[3,2-h]quinoline structure”,
11th Eurasia Conference
on Chemical Sciences, The Dead Sea (Jordan), October,
6th-10th, 2010. (P)
-
M. El-Abadelah, J. Zahra, S. Al-Trawneh,
P. Vicini, F. Zani. “Antibacterial and antitumor
activity of tetracyclic thienopyridones 4-Oxopyrido[3’,2’:
4,5]thieno[3,2-b] indoles”, 11th
Eurasia Conference on Chemical Sciences, The Dead Sea
(Jordan), October, 6th-10th, 2010. (P)
-
R.A. Al-Qawasmeh, J.A. Zahra, M.M.
El-Abadelah, R. Al-Bashiti, F. Zani, P. Vicini.
“Synthesis and antimicrobial activities
of some thiadiazolo-fused fluoroquinolones”,
11th Eurasia Conference
on Chemical Sciences, The Dead Sea (Jordan), October,
6th-10th, 2010. (P)
-
F. Zani, P. Vicini, A. Cavazzoni, S.
Al-Trawneh, J. Zahra, M. Kamal, M. El-Abadelah.
“Antibacterial and antitumor activity of
tetracyclic fluoroquinolones with pyrido[2,3-a]carbazole
structure”, 11th Eurasia
Conference on Chemical Sciences, The Dead Sea
(Jordan), October, 6th-10th, 2010.
(P)
-
P. Vicini, A.M. Panico, A. Geronikaki,
F. Zani, M. Incerti.
“Benzisothiazolylimino-5-benzylidene-4-thiazolidinones as
potential biologically active agents”,
11th Eurasia Conference
on Chemical Sciences, The Dead Sea (Jordan), October,
6th-10th, 2010. (P)
-
E. Moretti, S. Catinella, V. Mileo, C.
Silva, F. Vacondio, M. Mor. “MS
characterization of the catalytic domain of epidermal growth
factor receptor”, MASSA 2010 – 6th
MS Pharmaday, Milan (Italy), October, 6th-10th,
2010. (Poster Po-18). (P)
-
F. Vacondio, C. Silva, S. Rivara, M.
Mor, A. Bedini, G. Spadoni, G. Tarzia.
“Comparative in vitro metabolism of the
MT2-selective melatonin receptor ligands UCM765
and UCM924”, MASSA 2010 – 6th
MS Pharmaday, Milan (Italy), October, 6th-10th,
2010. (Poster Po-29). (P)
-
R. Menabeni, C. Scarpignato, R. Bettini.
“Sucralfate-anti-arthritic drug complex
formation in aqueous solution”, FIP
Pharmaceutical Sciences 2010 World Congress/AAPS Annual
Meeting and Exposition, New Orleans (Louisiana, USA),
November, 14th-18th, 2010.
(Poster #: T3114). (P)
-
L. Pezzini, F. Guida, R. Bettini.
“Phase behavior of diazepam-PEG binary
misture and stability of the relevant solid dispersions”,
FIP Pharmaceutical Sciences 2010
World Congress/AAPS Annual Meeting and Exposition,
New Orleans (Louisiana, USA), November, 14th-18th,
2010. (Poster #: T3121). (P)
-
C. Conti, A. Rossi, C. Carrisi, P.
Colombo. “A new assemled delivery
system of clrarithromycin and amoxicillin for helicobacter
pylori therapy”, FIP Pharmaceutical
Sciences 2010 World Congress/AAPS Annual Meeting and
Exposition, New Orleans (Louisiana, USA), November,
14th-18th, 2010. (P)
-
A.G. Balducci, P. Colombo, N. Khan, K.
Yuen, E. Magosso, G. Colombo, A. Rossi.
“Preparation of soft agglomerates based
on artemisinin-βCD complexes”,
FIP Pharmaceutical Sciences 2010
World Congress/AAPS Annual Meeting and Exposition,
New Orleans (Louisiana, USA), November, 14th-18th,
2010. (P).
-
M. Tognolini, C. Giorgio, I.H. Mohamed,
L. Flammini, M. Incerti, A. Lodola, E. Barocelli.
“Lithocholic acid competitively inhibits EphA2-ephrinA1
binding: pharmacological and structural considerations”,
22nd EORTC-NCI-AACR
Symposium on Molecular Targets and Cancer Therapeutics,
Berlin (Germany), November, 16th-19th,
2010. (Poster 293). (P)
-
S. Mercuri, P. Colombo.
“Assemblati modulari per una terapia orale multi-farmaco e
multi-cinetica del morbo di Parkinson”,
50° Simposio AFI, Rimini,
9-11 Giugno 2010. (C)
-
B.
RANIERI, M. GIORI, C. CURTI, L. BATTISTINI, F. ZANARDI, G.
CASIRAGHI. “Catalytic, Enantioselective
Vinylogous Mukaiyama-Mannich Reactions Exploiting Pyrrole-Based
Dienoxy Silanes”, XXXV “A. Corbella” Summer School,
Gargnano (BS), 14-18 Giugno 2010 (P)
-
A.M. Panico, P. Vicini, I. Crasci, M.
Incerti, G. Ronsisvalle.
“2-Benzisothiazolylimino-5-benzylidene-4-thiazolidinones as
MMP-13 inhibitors and antioxidant agents”,
XX National Meeting on Medicinal
Chemistry, Abano Terme (PD), 12-16 Settembre 2010.
(P)
-
A. Lodola, L. Capoferri, S.
Rivara, M. Mor, M. Mileni, A. Duranti, A. Tontini, G.
Tarzia, D. Piomelli, A.J. Mulholland.
“Chemical determinants of fatty acid
amide hydrolase inactivation explored by QM/MM mechanistic
modelling”, XX National Meeting on
Medicinal Chemistry, Abano Terme (PD), 12-16
Settembre 2010. (C)
-
C.
CURTI, B. RANIERI, L. BATTISTINI, F. ZANARDI, G.
CASIRAGHI. “Tuning the Reactivity of Silyloxy Pyrroles
towards Catalytic, Enantioselective Vinylogous Mukaiyama
Aldol and Mannich Processes”, XXXIII Convegno Nazionale
della Divisione di Chimica Organica della Società Chimica
Italiana, San Benedetto del Tronto (AP), 12-16 Settembre
2010 (C)
-
S. Sanchini, A. Duranti, A. Tontini, G.
Tarzia, A. Lodola, S. Rivara, F. Vacondio, M. Mor, J.R.
Clapper, G. Moreno-Sanz, D. Piomelli. “Scoperta del
primo inibitore dell’enzima idrolasi delle ammidi degli
acidi grassi (FAAH) ad azione periferica”,
10° SAYCS, Pesaro, 18-20
Ottobre 2010 (P)
-
B.
RANIERI. “Dienossi-silani eterociclici in reazioni
aldoliche viniloghe catalitiche ed enantioselettive”, XXV
Edizione “Nuovi Orientamenti nella Sintesi Organica”,
Milano, 15 Novembre 2010 (C)
-
F. Sonvico. “Preparazioni
solide orali per la somministrazione di farmaci combinati in
una sola forma di dosaggio”, Workshop Next Generation
Medicines, Bologna, 30 Novembre 2010. (C)
IV. Invited
speakers
-
P. Colombo.
“Combination products and innovation in drug delivery
systems”,
Incontro in Merck KGaA,
Darmstadt (Germany), February, 17th,
2010.
-
R. Bettini.
“Supercritical fluids in modern drug delivery for particle
and crystal engineering”, One Day
Seminar Drug Delivery Strategies for Infectoious diseases,
Universiti Sains Malaysia, Penang (Malaysia), February, 24th,
2010.
-
O.L. Strusi, F. Sonvico, P. Barata, S.
Mercuri, G. Colombo, F. Buttini, R. Bettini, P. Colombo.
“Multi-kinetics and site-specific oral delivery system of
artesunate-clindamycin combination for malaria treatment”,
7th World Meeting on
Pharmaceutics, Biopharmaceutics and Pharmaceutical
Technology, La Valletta (Malta), March, 8th-11th,
2010.
-
R. Bettini.
“Water as activating agent in swelling controller drug
delivery systems”, Frontiers in
water biophysics, Trieste (Italy), May, 23th-26th,
2010.
-
P. Colombo.
“Dome Matrix technology and application in malaria”,
Pharmatech 2010, International
Conference and Exhibition on Pharmaceutical, Nutraceutical
and Cosmeceutical Technology, Kuala Lumpur
(Malaysia), May, 25th-27th, 2010.
-
G. Costantino.
“Searching for new antipsychotic drugs. When the target is
complex (or a complex is the target)”,
Workshop in Medicinal Chemistry and
Complex Systems: New Opportunities for Rational Drug Design,
Parma (Italy), June, 4th, 2010.
-
P. Colombo.
“Dry powder inhalers: construction of antibiotic
microparticles for lung infection treatment”,
Third International Meeting on
Pharmacy & Pharmaceutical Sciences, Istanbul
(Turkey), June 9th, 2010.
-
A. Lodola.
IV Conference on
Modeling and Design of Molecular Materials 2010,
Wroclaw (Poland), July 4th-8th, 2010.
-
S. Nicoli.
“Drug delivery: an overview”,
Summer School on
Pharmaceutical Analysis (SSPA),
Rimini, Italia, June 13th-16th 2010.
-
R. Bettini.
“Polimorphs in supercritical processes: a pharmaceutical
prospect”, 5th Bologna
Convention on Crystal form, Bologna (Italy),
September, 1st-4th, 2010.
-
P. Colombo.
“Multi-kinetics and site-specific oral delivery system for
malaria treatment”, 15th
International Pharmaceutical Symposium, Antalya
(Turkey), September, 13th-15th, 2010.
-
P. Colombo.
“Novel platforms for oral drug delivery”,
Advances in Pharmacotherapy,
Trento (Italy), September, 24th, 2010.
-
R. Bettini.
“Smoothed lactose carriers”, Meeting
on Lactose as a Carrier for Inhalation Products,
Parma (Italy), September 26th-28th,
2010. (C)
-
S. Nicoli.
“Trans-scleral delivery of macromolecules: the iontophoretic
approach”,
2nd Conference on “Innovation
in drug delivery: from preformulation to development through
innovative evaluation process”,
Aix-en-Provence, Francia, October 3th-6th,
2010.
-
P. Colombo.
“Dome Matrix Technology: the assemblage of modules for oral
delivery of combined drugs”, CPhI
worldwide 2010, Paris (France), October, 5th-7th,
2010.
-
A. Lodola.
“Application of computetional methods to the design of
enzyme inhibitors”, BioReC, School
of Life Sciences, Northumbria University, Newcastle
(U.K.), October 22nd, 2010.
-
P. Colombo.
“Pharmaceutics and formulation of nutraceuticals,
traditional medicines and phytopharmaceuticals”,
International Conference on Natural
Products, Penang (Malaysia), December, 10th-12th,
2010.
-
P. Colombo.
“Pulmonary systems”, Third Biotech
Workshop Drug delivery systems for biotech products,
Pavia, 24-25 Marzo 2010.
-
P. Colombo. “Rapporti fra
Università ed aziende per lo sviluppo di nuove tecnologie”,
Seminario “Il contract manufacturing
oggi in Italia” nell’ambito della mostra Pharmintech,
Bologna, 12-14 Maggio 2010.
-
P. Colombo. “Ricerca, terapia,
impatto economico: tre approcci diversi alla sfida delle
medicine personalizzate”, Le
medicine personalizzate tra prospettive scientifiche e
necessità di governo clinico, Università degli Studi
di Parma, Parma, 12 Ottobre 2010.
-
P. Colombo. “Swelling activated
multi-kinetics and site-specific oral drug delivery systems”,
Giornata in memoria della Prof.ssa
Maria Edvige Sangalli: Advanced Drug Delivery Systems,
Milano, 2 Novembre 2010.
-
P. Colombo.
“Consorzio Tefarco:positiva esperienza di un network”,
Workshop “Know how sarin: a way to
effective and efficient research?”, Sala Congressi
Azienda Ospedaliero-Universitaria di Parma, Parma, 22
Novembre 2010.
V. Chairperson
-
P.
Colombo.
7th World Meeting on
Pharmaceutics, Biopharmaceutics and Pharmaceutical
Technology, La Valletta (Malta), March, 8th-11th,
2010.
-
M. MOR .
Workshop in
Medicinal Chemistry and Complex Systems: New
Opportunities for Rational Drug Design,
Parma (Italy), June, 4th, 2010.
VI. Awards
-
P. Colombo.
Doctor Honoris Causa della Faculty of Pharmacy della
National and Kapodistrian University of Athens, Athens
(Greece), April 22nd, 2010.
-
A. Lodola.
Runner-up of the EFMC Prize for a Young Medicinal Chemist in
Academia, Brussels, September 5th-9th,
2010.
-
P. Colombo. Elezione a Preside
della Facoltà di Farmacia del Dipartimento Farmaceutico
dell’Università degli Studi di Parma per il quadriennio
2010-2014.
-
P. Colombo. Membro esperto della
European Medicines Agency (EMEA).
-
A. Rossi. Professeur Invitée
presso la Faculté de Medicine et Pharmacie dell’Université
Claude Bernard - Lyon 1 (France) per i periodi 18 Aprile
2010 – 1° Maggio 2010 e 20 Giugno 2010 – 3 Luglio 2010.
-
C. Conti. Travel award dalla
European Federation for Pharmaceutical Sciences (EUFEPS) per
partecipare al 2010 FIP PSWC/AAPS Annual Meeting and
Exposition a New Orleans (Louisiana, USA), November 14th.18th,
2010.
-
B.
RANIERI. Premio di Laurea conferito dal Gruppo
Interdivisionale di Catalisi (GIC) della SCI in occasione
della XXV Edizione “Nuovi Orientamenti nella Sintesi
Organica”, Milano, 15 Novembre 2010.
-
P. Vicini, M. Incerti. Premio
“Bioorganic & Medicinal Chemistry Most Cited Articles 2003
to 2010” per l’articolo scientifico di P. Vicini, A.
Geronikaki, M. Incerti, B. Busonera, G. Poni, C.A. Cabras,
P. La Colla: “Synthesis and biological evaluation of benzo[d]isothiazole,
benzothiazole and thiazole Schiff bases” pubblicato sulla
rivista Bioorganic and Medicinal Chemistry, Volume 11(22),
pagine 4785-4789 (2003).
VII. Visiting
researchers
-
Stefania Aiello, Università di
Palermo, Facoltà di Farmacia, 01.02.2009 – 31.01.2010.
-
Faisalina Bt Ahmad Fisol,
Pumpong, Malaysia, 27.10.2009 – 15.01.2010.
VIII. Visiting
students
-
Paulo Renato
Oliveira, Universidade
Federal de Santa Catarina, Brasile, 13.09.2009 – 13.02.2010.
-
Ayse Gosku Kaya,
University of Ankara, Turkey, 01.10.2009 – 28.02.2010.
-
Tengku Fahima Azira
Tuan Mat, Kota Bharu,
Malaysia, 18.01.2010 – 23.03.2010.
-
Flavia Almada Do
Carmo, Laboratório de
Tecnologia Industrial Farmacêutica, Departamento de
Medicamentos Faculdade de Farmácia, Universidade Federal do
Rio de Janeiro, Brasile, 19.05.2010 – 30.04.2011.
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